Yayınlar & Eserler

SCI, SSCI ve AHCI İndekslerine Giren Dergilerde Yayınlanan Makaleler

Development of Thiazolidinones as Fungal Carbonic Anhydrase Inhibitors.

International journal of molecular sciences, cilt.21, 2020 (SCI Expanded İndekslerine Giren Dergi) identifier identifier

Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold.

Journal of enzyme inhibition and medicinal chemistry, cilt.34, ss.1400-1413, 2019 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies.

Journal of enzyme inhibition and medicinal chemistry, cilt.34, ss.1051-1061, 2019 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

Novel 2-indolinones containing a sulfonamide moiety as selective inhibitors of candida β-carbonic anhydrase enzyme.

Journal of enzyme inhibition and medicinal chemistry, cilt.34, ss.528-531, 2019 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

Aromatase inhibition by 2-methyl indole hydrazone derivatives evaluated via molecular docking and in vitro activity studies.

Xenobiotica; the fate of foreign compounds in biological systems, cilt.49, ss.549-556, 2019 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

Novel sulfonamide-containing 2-indolinones that selectively inhibit tumor-associated alpha carbonic anhydrases.

Bioorganic & medicinal chemistry, cilt.25, ss.3714-3718, 2017 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

Target Recognition Molecules and Molecular Modeling Studies

Current Topics In Medicinal Chemistry, cilt.17, ss.1580-1587, 2017 (SCI Expanded İndekslerine Giren Dergi)

Isatin analogs as novel inhibitors of Candida spp. β-carbonic anhydrase enzymes.

Bioorganic & medicinal chemistry, cilt.24, ss.1648-52, 2016 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

A Divalent PAMAM-Based Matrix Metalloproteinase/Carbonic Anhydrase Inhibitor for the Treatment of Dry Eye Syndrome.

Chemistry (Weinheim an der Bergstrasse, Germany), cilt.22, ss.1714-21, 2016 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives.

European journal of medicinal chemistry, cilt.107, ss.82-96, 2016 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

Computational investigation of the selectivity of salen and tetrahydrosalen compounds towards the tumor-associated hCA XII isozyme.

Journal of enzyme inhibition and medicinal chemistry, cilt.30, ss.114-8, 2015 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

Fragment growing induces conformational changes in acetylcholine-binding protein: a structural and thermodynamic analysis.

Journal of the American Chemical Society, cilt.133, ss.5363-71, 2011 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

A G(q/11)-coupled mutant histamine H(1) receptor F435A activated solely by synthetic ligands (RASSL).

The Journal of biological chemistry, cilt.280, ss.34741-6, 2005 (SCI Expanded İndekslerine Giren Dergi) identifier identifier identifier

Hakemli Kongre / Sempozyum Bildiri Kitaplarında Yer Alan Yayınlar

Computer Aided Design and Synthesis of New Ursane Triterpenoids with Nuclear Factor Kappa B Inhibition Effect

7th International BAU Drug Design Congress, İstanbul, Türkiye, 19 - 21 December 2019, ss.159-160 Creative Commons License

The application of molecular modelling studies to understand the selectivity and potency of several novel carbonic anhydrase inhibitors

the 4th International Satellite Meeting on Carbonic Anhydrase, Parma, İtalya, 14 - 17 November 2019

Molecular docking and in vitro bioactivity of 5-fluoroindole derivatives on ER, aromatase and CYP1B1 activity in breast cancer cells

55th Congress of the European-Societies-of-Toxicology (EUROTOX) - Toxicology - Science Providing Solutions, Helsinki, Finlandiya, 8 - 11 September 2019, cilt.314

Hit Identification Against DNA Topoisomerases Using Virtual Screenings

7. uluslararası ilaç kimyası kongresi, Antalya, Türkiye, 14 - 17 March 2019

Bazı Uvaol Türevlerinin Sentezi ve in vitro Biyoaktivitelerininİncelenmesi

3rd International Convention of Pharmaceuticals and Pharmacies, İstanbul, Türkiye, 26 April 2017, ss.580-581 Creative Commons License

Bazı Uvaol Türevlerinin Sentezi ve in vitro Biyokaitivitelerininİncelenmesi

IVEK 3rd International Convention of Pharmaceuticals and Pharmacies3. Uluslararası İlaç ve Eczacılık Kongresi, İstanbul., 26 April - 29 January 2017

Nükleer Faktör Kappa-B İnhibisyon Etkili Ursan Türevi Triterpenlerin Sentezi

Uluslararası Katılımlı 5. İlaç Kimyası: İlaç Etkin Maddesi Tasarımı, Sentezi, Üretimi ve Standardizasyonu Kongresi, Antalya, Türkiye, 30 March - 02 April 2017, ss.131 Creative Commons License

Structurally novel isatin derivatives as putative anticancer and antifungal agents

7th European Congress of Pharmacology (EPHAR2016), İstanbul, Türkiye, 01 July 2016, ss.1

Bilgisayar-destekli Antikolinesteraz 3-Hidroksiflavon Türevlerinin Sentezi ve in vitro Aktivite Çalışmaları.

2. Bilgisayar Destekli İlaç Tasarımı Kursu (Uygulamalı), İstanbul, Türkiye, 16 May 2016, ss.163

Molecular modelling studies to understand the effects of bioactive compounds on DNA and gene expression

TURKHELTOX Toxicology Congress, 9th Congress of the Turkish Society of Toxicology with participation of the Hellenic Society of Toxicology, İzmir, Türkiye, 21 November 2015, ss.1

The Search for Novel 3-hydroxyflavones with Anticholinergic Activity.

Royal Society of Chemistry, Medicinal Chemistry Residential School, Loughbrough, İngiltere, 11 June 2015, ss.232

Docking studies to investigate ligand-protein binding interactions in pharmaceutically important carbonic anhydrases

10th international carbonic anhydrase conference, Maastricht, Hollanda, 12 May 2015, ss.1

Abietane diterpenoids as butyrylcholinesterase inhibitors from Salvia species

International Congress on Natural Products Research on Global Change, Natural Products and Human Health/8th Joint Meeting of AFERP, ASP, GA, PSE and SIF, New-York, Amerika Birleşik Devletleri, 28 July - 01 August 2012, cilt.78, ss.1229

Potent inhibitors of mitochondrial carbonic anhydrase isozymes CA-VA and CA-VB and brain-associated CA-VII

9th International conference on Carbonic Anhydrases (CA), İstanbul, Türkiye, 11 April 2012, ss.1

The quest for nicotinic receptor ligands by using AChBP as a template

XIXst International Symposium on Medicinal Chemistry, İstanbul, Türkiye, 29 August 2006, ss.25

Kitap & Kitap Bölümleri

Carbonic Anhydrases as Biocatalysts: From Theory to Medical and Industrial Applications

Chapter 7. The structure, physiological role and potential medicinal applications of Carbonic Anhydrase V, G. De Simone & C.T. Supuran, Editör, Elsevier Science, Oxford/Amsterdam , Waltham, ss.125-138, 2015

Pharmacology of nicotinic acetylcholine receptors from the basic and therapeutic perspectives

Chapter 3. The acetylcholine binding protein as a template for the ligand binding domains of the homologous nicotinic receptors, Hugo R. Arias, Editör, Research Signpost, Kerala, ss.45-70, 2011