Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold.


Rotondi G., Guglielmi P., Carradori S., Secci D., De Monte C., De Filippis B., ...More

Journal of enzyme inhibition and medicinal chemistry, vol.34, pp.1400-1413, 2019 (SCI-Expanded) identifier identifier identifier

  • Publication Type: Article / Article
  • Volume: 34
  • Publication Date: 2019
  • Doi Number: 10.1080/14756366.2019.1651315
  • Journal Name: Journal of enzyme inhibition and medicinal chemistry
  • Journal Indexes: Science Citation Index Expanded (SCI-EXPANDED), Scopus
  • Page Numbers: pp.1400-1413
  • Keywords: Carbonic anhydrase inhibitor, sulfoxide enantioseparation, carboxylic acid, molecular modelling, CARBONIC-ANHYDRASE-IX, FASCINATING MOLECULAR FRAMEWORK, ENANTIOSEPARATION ABILITY, SULFONAMIDE DERIVATIVES, DRUG DISCOVERY, CANCER, PH, 3-(PHENYL-4-OXY)-5-PHENYL-4,5-DIHYDRO-(1H)-PYRAZOLE, ENANTIOMERS, ASSIGNMENT
  • Bezmialem Vakıf University Affiliated: Yes