Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors.


Güzel-Akdemır Ö., Angelı A., Demır K., Supuran C., Akdemir A.

Journal of enzyme inhibition and medicinal chemistry, cilt.33, ss.1299-1308, 2018 (SCI-Expanded, Scopus) identifier identifier identifier

  • Yayın Türü: Makale / Tam Makale
  • Cilt numarası: 33
  • Basım Tarihi: 2018
  • Doi Numarası: 10.1080/14756366.2018.1499628
  • Dergi Adı: Journal of enzyme inhibition and medicinal chemistry
  • Derginin Tarandığı İndeksler: Science Citation Index Expanded (SCI-EXPANDED), Scopus
  • Sayfa Sayıları: ss.1299-1308
  • Anahtar Kelimeler: carbonic anhydrase IX, hCA IX, thiazolidinone, molecular modelling, docking, TARGETING TUMOR HYPOXIA, BIOLOGICAL EVALUATION, SELECTIVE INHIBITORS, DERIVATIVES, POTENT, XII, AGENTS, 4-THIAZOLIDINONE, ANTIFUNGAL, ISOZYMES
  • Bezmiâlem Vakıf Üniversitesi Adresli: Evet