Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies.


Ammazzalorso A., Carradorı S., Angelı A., Akdemir A., De Filippis B., Fantacuzzı M., ...Daha Fazla

Journal of enzyme inhibition and medicinal chemistry, cilt.34, ss.1051-1061, 2019 (SCI-Expanded, Scopus) identifier identifier identifier

  • Yayın Türü: Makale / Tam Makale
  • Cilt numarası: 34
  • Basım Tarihi: 2019
  • Doi Numarası: 10.1080/14756366.2019.1611801
  • Dergi Adı: Journal of enzyme inhibition and medicinal chemistry
  • Derginin Tarandığı İndeksler: Science Citation Index Expanded (SCI-EXPANDED), Scopus
  • Sayfa Sayıları: ss.1051-1061
  • Anahtar Kelimeler: N-acylsulphonamides, carbonic anhydrase, PPAR antagonist, fibrate derivatives, benzothiazole, benzophenone, SECONDARY SULFONAMIDES, ISOFORMS I, ISOZYME-II, SELECTIVE-INHIBITION, DRUG DISCOVERY, XII, BINDING, ACYLSULFONAMIDES, VITRO, BENZENESULFONAMIDES
  • Bezmiâlem Vakıf Üniversitesi Adresli: Evet