Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies.


Ammazzalorso A., Carradorı S., Angelı A., Akdemir A., De Filippis B., Fantacuzzı M., ...More

Journal of enzyme inhibition and medicinal chemistry, vol.34, pp.1051-1061, 2019 (SCI-Expanded) identifier identifier identifier

  • Publication Type: Article / Article
  • Volume: 34
  • Publication Date: 2019
  • Doi Number: 10.1080/14756366.2019.1611801
  • Journal Name: Journal of enzyme inhibition and medicinal chemistry
  • Journal Indexes: Science Citation Index Expanded (SCI-EXPANDED), Scopus
  • Page Numbers: pp.1051-1061
  • Keywords: N-acylsulphonamides, carbonic anhydrase, PPAR antagonist, fibrate derivatives, benzothiazole, benzophenone, SECONDARY SULFONAMIDES, ISOFORMS I, ISOZYME-II, SELECTIVE-INHIBITION, DRUG DISCOVERY, XII, BINDING, ACYLSULFONAMIDES, VITRO, BENZENESULFONAMIDES
  • Bezmialem Vakıf University Affiliated: Yes